Zaloguj się
dr Dawid Warszycki
dr Dawid Warszycki
+48 12 6623301
warszyc@if-pan.krakow.pl
pokój 326 
Zakład Chemii LekówDokonania naukowe
- Publikacje
Novel Tripeptides as Tyrosinase Inhibitors: In Silico and In Vitro Approaches
Autorzy: Michał Dymek, Dawid Warszycki, Sabina Podlewska, Elżbieta Sikora
DOI: 10.3390/ijms252413509
Date: 2024-12-17
Isomeric Activity Cliffs—A Case Study for Fluorine Substitution of Aminergic G Protein-Coupled Receptor Ligands
Autorzy: Wojciech Pietruś, Rafał Kurczab, Dawid Warszycki, Andrzej J. Bojarski, Jürgen Bajorath
DOI: 10.3390/molecules28020490
Date: 2023-01-04
Improved HDAC Inhibition, Stronger Cytotoxic Effect and Higher Selectivity against Leukemias and Lymphomas of Novel, Tricyclic Vorinostat Analogues
Autorzy: Bartosz Bieszczad, Damian Garbicz, Marta Świtalska, Marta K. Dudek, Dawid Warszycki, Joanna Wietrzyk, Elżbieta Grzesiuk, Adam Mieczkowski
DOI: 10.3390/ph14090851
Date: 2021-08-26
Novel Vorinostat Analogues with Improved HDAC Inhibition, Stronger Cytotoxic Effect and Higher Selectivity Against Leukemias and Lymphomas
Autorzy: Bartosz Bieszczad, Damian Garbicz, Marta Świtalska, Marta K. Dudek, Dawid Warszycki, Joanna Wietrzyk, Elżbieta Grzesiuk, Adam Mieczkowski
DOI: 10.20944/preprints202105.0251.v1
Date: 2021-05-11
Design, synthesis and biological evaluation of 2-substituted-6-[(4-substituted-1-piperidyl)methyl]-1H-benzimidazoles as inhibitors of ebola virus infection
Autorzy: Maxime Bessières, Elżbieta Plebanek, Payel Chatterjee, Punya Shrivastava-Ranjan, Mike Flint, Christina F. Spiropoulou, Dawid Warszycki, Andrzej J. Bojarski, Vincent Roy, Luigi A. Agrofoglio
DOI: 10.1016/j.ejmech.2021.113211
Date: 2021-03-01
Rationally designed N-phenylsulfonylindoles as a tool for the analysis of the non-basic 5-HT<sub>6</sub>R ligands binding mode.
Autorzy:
DOI: 10.1016/j.ejmech.2020.112916
Date: 2020-10-09
Virtual screening-driven discovery of dual 5-HT<sub>6</sub>/5-HT<sub>2A</sub> receptor ligands with pro-cognitive properties.
Autorzy:
DOI: 10.1016/j.ejmech.2019.111857
Date: 2019-11-07
In Silico Methods for the Discovery of Orthosteric GABA<sub>B</sub> Receptor Compounds
Autorzy: Linn M. Evenseth, Dawid Warszycki, Andrzej Bojarski, Mari Gabrielsen, Ingebrigt Sylte
DOI: 10.3390/molecules24050935
Date: 2019-03-01
The effect of the intramolecular C-H⋯O interactions on the conformational preferences of bis-arylsulfones-5-HT<inf>6</inf>receptor antagonists and beyond
Autorzy: Kalinowska-Tłuścik, J., Staroń, J., Krawczuk, A., Mordalski, S., Warszycki, D., Satała, G., Hogendorf, A.S., Bojarski, A.J.
DOI: 10.1039/c8ra03107j
Date: 2018-01-01
Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs
Autorzy: Tber, Z., Wartenberg, M., Jacques, J.-E., Roy, V., Lecaille, F., Warszycki, D., Bojarski, A.J., Lalmanach, G., Agrofoglio, L.A.
DOI: 10.1016/j.bmc.2018.07.032
Date: 2018-01-01
